北京师范大学放射性药物教育部重点实验室
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贾红梅


教授,博士生导师,理学博士(北京师范大学),德国莱比锡多学科综合同位素研究院访问学者和高级访问学者,德国亥姆霍兹Dresden-Rossendorf研究中心放射性药物癌症研究院高级研究学者。

通信地址:北京市新街口外大街19号 北京师范大学化学学院

邮编:100875

电话:010 5880 8891

传真:010 5880 8891

电子邮箱:hmjia@bnu.edu.cn


讲授课程


放射性药物化学,普通化学实验。


研究兴趣


放射性药物化学,生物功能显像分子探针的研究。


主持的科研项目


1. 用于肿瘤诊断和个性化治疗的Tc-99m/Re-188标记的s2受体放射性药物研究,2015.1−2018.12,国家自然科学基金项目(21471019);

2. Tc-99m标记的s2受体肿瘤分子探针的研究,2010.1−2013.12,国家自然科学基金项目(21071023);
3. Tc-99m标记的s受体肿瘤显像剂的研究,2006.1−2008.12,国家自然科学基金项目(20501004);
4. 还原醚化反应及其在F-18标记的PET放射性药物合成中的应用研究,教育部留学回国人员科研启动基金;
5. 肿瘤显像与治疗,2013.4−2013.10,国家自然科学基金国际合作与交流项目(21310102012);
6. Sigma受体分子探针的研究,2011.10−2011.11,国家自然科学基金国际合作与交流项目(21110102042);
7. Sigma受体显像剂的研究,2008.10.19−2008.10.26,国家自然科学基金国际合作与交流项目(20810102039);
8. Sigma受体显像剂的生物评价方法,2007.10,国家自然科学基金国际合作与交流项目。

代表性论文


1. Li Dan, Chen Yuanyuan, Wang Xia, Deuther-Conrad Winnie, Chen Xin , Jia Bing, Dong Chengyan, Steinbach Jörg, Brust Peter, Liu Boli, Jia Hongmei*. 99mTc-cyclopentadienyl tricarbonyl chelate-labeled compounds as selective sigma-2 receptor ligands for tumor imaging. Journal of Medicinal Chemistry, 2016, 59(3): 934-946.

2. Xie Fang, Bergmann Ralf, Kniess Torsten, Deuther-Conrad Winnie, Mamat Constantin, Neuber Christin, Liu Boli, Steinbach Jörg, Brust Peter, Pietzsch Jens, Jia Hongmei*.18F-labeled 1,4-dioxa-8-azaspiro[4.5]decane derivative: synthesis and biological evaluation of a s1 receptor radioligand with low lipophilicity as potent tumor imaging agent. Journal of Medicinal Chemistry, 2015, 58(14), 5395-5407.
3. Wang Xia, Li Dan, Deuther-Conrad Winnie, Lu Jie, Xie Ying, Jia Bing, Cui Mengchao, Steinbach Jörg, Brust Peter, Liu Boli, Jia Hongmei*. Novel cyclopentadienyl tricarbonyl 99mTc complexes containing 1-piperonylpiperazine moiety: potential imaging probes for sigma-1 receptors. Journal of Medicinal Chemistry, 2014, 57(16), 7113-7125.
4. Li Yan, Wang Xia, Zhang Jinming, Deuther-Conrad Winniw, Xie Fang, Zhang Xiaojun, Liu Jian, Qiao Jinping, Cui Mengchao, Steinbach Joerg, Brust Peter, Liu Boli, Jia Hongmei*. Synthesis and evaluation of novel 18F-labeled spirocyclic piperidine derivatives as σ1 receptor ligands for positron emission tomography imaging. Journal of Medicinal Chemistry, 2013, 56(9), 3478-3491.
5. Xie Fang, Kniess Torsten, Neuber Christin, Deuther-Conrad Winnie, Mamat Constantin, Lieberman Brian P., Liu Boli, Mach Robert H., Brust Peter, Steinbach Jörg, Pietzsch Jens, Jia Hongmei*. Novel indole-based sigma-2 receptor ligands: synthesis, structure–affinity relationship and antiproliferative activity. Med. Chem. Commun., 2015, 6, 1093-1103.
6. Chen Yuan-Yuan, Wang Xia , Zhang Jin-Ming, Deuther-Conrad Winnie, Zhang Xiao-Jun, Huang Yiyun, Li Yan, Ye Jia-Jun, Cui Meng-Chao, Steinbach Joerg, Brust Peter, Liu Bo-Li, Jia Hong-Mei*. Synthesis and evaluation of a 18F-labeled spirocyclic piperidine derivative as promising s1 receptor imaging agent. Bioorganic & Medicinal Chemistry 2014, 22: 5270–5278.
7. Wang Xia, Li Yan, Deuther-Conrad Winnie, Xie Fang, Chen Xin, Cui Meng-Chao, Zhang Xiao-Jun, Zhang Jin-Ming, Steinbach Jörg, Brust Peter, Liu Bo-Li, Jia Hong-Mei*. Synthesis and biological evaluation of 18F labeled fluoro-oligo-ethoxylated 4-benzylpiperazine derivatives for sigma-1 receptor imaging. Bioorganic & Medicine Chemistry 2013, 21: 215-222.
8. Chen Xin, Cui Meng-Chao, Deuther-Conrad Winnie, Tu Ying-Feng, Ma Teng, Xie Ying, Jia Bing, Li Yan, Xie Fang, Wang Xia, Steinbach Jörg, Brust Peter, Liu Bo-Li, Hong-Mei Jia*. Synthesis and biological evaluation of a novel 99mTc cyclopentadienyl tricarbonyl complex ([(Cp-R)99mTc(CO)3]) for sigma-2 receptor tumor imaging. Bioorganic & Medicinal Chemistry Letters 2012, 22: 6352-6357.
9. Li Zi-jing, Ren Hui-Ying, Cui Meng-Chao, Deuther-Conrad Winnie, Tang Rui-Kun, Steinbach Jörg, Brust Peter, Liu Bo-Li, Jia Hong-Mei*. Synthesis and biological evaluation of novel 4-benzylpiperazine ligands for sigma-1 receptor imaging. Bioorganic & Medicinal Chemistry 2011, 19: 2911-2917.
10. Jia Hong-Mei, Fang De-Cai*, Scheunemann Matthias. Theoretical studies on reductive etherification reactions between aromatic aldehydes and alcohols. Journal of Organic Chemistry 2005, 70(11): 4478-4483.
 

 

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