北京师范大学放射性药物教育部重点实验室
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2014年科研论文汇总
发布时间: 2015-01-12
 

 

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SCI/EI/国内期刊

论文作者

1

One-Dimensional Channels Encapsulated in Supramolecular Networks Constructed of Zinc(II), Manganese(II), or Nickel(II) Atoms with 3-(Carboxymethyl)-2,7-dimethyl-3H-benzo[d]imidazole-5-carboxylic Acid

ZEITSCHRIFT FUR ANORGANISCHE UND ALLGEMEINE CHEMIE

2014, 640(1): 159-167

SCI

Zhao, Mingxia; Xiong, Liqin; Li, Shilei; Chang, Jin; Ning, Hongyu; Qi, Chuanmin

2

Tc-99m-labeled benzothiazole and stilbene derivatives as imaging agents for A beta plaques in cerebral amyloid angiopathy

MEDCHEMCOMM

2014, 5(2): 153-158

SCI

Jia, Jianhua; Cui, Mengchao; Dai, Jiapei; Wang, Xuedan; Ding, Yu-Shin; Jia, Hongmei; Liu, Boli

3

Past and Recent Progress of Molecular Imaging Probes for beta-Amyloid Plaques in the Brain

CURRENT MEDICINAL CHEMISTRY

2014, 21(1): 82-112

SCI

Cui, Mengchao

4

Molecular Imaging of alpha(1) Receptors In Vivo: Current Status and Perspectives

CURRENT MEDICINAL CHEMISTRY

2014, 21(1): 35-69

SCI

Brust, P.; Deuther-Conrad, W.; Lehmkuhl, K.; Jia, H.; Wuensch, B.

5

Radiolabeled Glucose Derivatives for Tumor Imaging Using SPECT and PET

CURRENT MEDICINAL CHEMISTRY

2014, 21(1): 24-34

SCI

Liu, T.; Zhang, J.; Wang, X.; Yang, J.; Tang, Z.; Lu, J.

6

Current Status and Progress of Radiopharmaceuticals for Molecular Imaging and Targeted Therapy

CURRENT MEDICINAL CHEMISTRY

2014, 21(1): 2-3

SCI

Zhang, Junbo

7

Combined 3D-QSAR, Molecular Docking, Molecular Dynamics Simulation, and Binding Free Energy Calculation Studies on the 5-Hydroxy-2H-Pyridazin-3-One Derivatives as HCV NS5B Polymerase Inhibitors

CHEMICAL BIOLOGY & DRUG DESIGN

2014,83(1): 89-105

SCI

Yu, Haijing; Fang, Yu; Lu, Xia; Liu, Yongjuan; Zhang, Huabei

8

Preparation and biological evaluation of (TcN)-Tc-99m-labeled pteroyl-lys derivative as a potential folate receptor imaging agent

JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS

2014, 57(1): 12-17

SCI

Chen, Yuan; Guo, Hongjuan; Xie, Fang; Lu, Jie

9

Neuroprotective Effects of Jitai Tablet, a Traditional Chinese Medicine, on the MPTP-Induced Acute Model of Parkinson's Disease: Involvement of the Dopamine System

EVIDENCE-BASED COMPLEMENTARY AND ALTERNATIVE MEDICINE

2014, 542383

SCI

Liu, Jia; Gao, Jinlong; Tu, Shaoang; Xu, Shasha; Liu, Ying; Shang, Weihu; Gu, Chenxin; Huang, Yiyun; Han, Mei

10

Pharmacokinetics and Biotransformation of Tea Polyphenols

CURRENT DRUG METABOLISM

2014, 15(1): 30-36

SCI

Qiao, Jinping; Kong, Xiangyi; Kong, Aiying; Han, Mei

11

Novel Tc-99m radiolabeled folate complexes with PEG linkers for FR-positive tumor imaging: synthesis and biological evaluation

RSC ADVANCES

2014, 4(61): 32197-32206

SCI

Xie, Fang; Zhang, Chun; Yu, Qian; Pang, Yan; Chen, Yuan; Yang, Wenjiang; Xue, Jingquan; Liu, Yu; Lu, Jie

12

PET/SPECT imaging agents for neurodegenerative diseases

CHEMICAL SOCIETY REVIEWS

2014,43(19): 6683-6691

SCI

Zhu, Lin; Ploessl, Karl; Kung, Hank F.

13

Evaluation of molecules based on the electron donor-acceptor architecture as near-infrared beta-amyloidal-targeting probes

CHEMICAL COMMUNICATIONS

2014, 50(80): 11875-11878

SCI

Fu, Hualong; Cui, Mengchao; Tu, Peiyu; Pan, Ziwei; Liu, Boli

14

Catalytic asymmetric Diels-Alder reactions involving aryl vinyl ketones

CHEMICAL COMMUNICATIONS

2014, 50(91): 14113-14116

SCI

Kong, Liman; Han, Xiaoyu; Jiao, Peng

15

The Interactions of Anticancer Agents with Tea Catechins: Current Evidence from Preclinical Studies

ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY

2014, 14(10): 1343-1350

SCI

Shang, Weihu; Lu, Weidong; Han, Mei; Qiao, Jinping

16

Synthesis and biological evaluation of fatty acids conjugates bearing cyclopentadienyl-donors incorporated [Tc-99m/Re(CO)(3)](+) for myocardical imaging

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

2014, 72, 10-17

SCI

Zeng, Huahui; Zhang, Huabei

17

Carbon-11 labeled stilbene derivatives from natural products for the imaging of A beta plaques in the brain

RADIOCHIMICA ACTA

2014, 102, 185-192

SCI

Cui, Mengchao; Tang, Ruikun; Zhang, Jinming; Zhang, Xiaojun; Li, Zijing; Jia, Hongmei; Liu, Boli

18

Radiopharmaceuticals in China: current status and prospects

RADIOCHIMICA ACTA

2014, 102, 53-67

SCI

Jia, Hong-Mei; Liu, Bo-Li

19

Receptor and ligand-based 3D-QSAR study on a series of pyrazines/pyrrolidylquinazolines as inhibitors of PDE10A enzyme

MEDICINAL CHEMISTRY RESEARCH

2014, 23(2):

775-789

SCI

Liu, Yongjuan; Lu, Xia; Xue, Tian; Hu, Shiyuan; Zhang, Huabei

20

Smart Near-Infrared Fluorescence Probes with Donor-Acceptor Structure for in Vivo Detection of beta-Amyloid Deposits

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

2014, 136(9): 3388-3394

SCI

Cui, Mengchao; Ono, Masahiro; Watanabe, Hiroyuki; Kimura, Hiroyuki; Liu, Boli; Saji, Hideo

21

Design of novel focal adhesion kinase inhibitors using 3D-QSAR and molecular docking

MEDICINAL CHEMISTRY RESEARCH

2014, 23(4): 1976-1997

SCI

Lu, Xia; Zhao, Lingzhou; Xue, Tian; Zhang, Huabei

22

SPECT imaging of dopamine transporter in heroin abusers with Jitai tablets maintenance treatment up to one year

JOURNAL OF NUCLEAR MEDICINE

2014, 55

SCI

Xu, Shasha; Liu, Ying; Lv, Rongbin; Wang, Yuankai; Yuan, Jie; Shang, Weihu; Han, Mei; Liu, Xingdang

23

SPECT imaging of dopamine transporter in heroin abusers with Jitai tablets maintenance treatment up to one year

JOURNAL OF NUCLEAR MEDICINE

2014, 55

SCI

Xu, Shasha; Liu, Ying; Lv, Rongbin; Wang, Yuankai; Yuan, Jie; Shang, Weihu; Han, Mei; Liu, Xingdang

24

Automated synthesis of novel F-18-labeled diarylideneacetone derivatives for in vivo imaging of beta-amyloid plaque

JOURNAL OF NUCLEAR MEDICINE

2014, 55

SCI

Li, Zijing; Kamble, Rajesh; Cui, Mengchao; Kothari, Paresh; Vallabhajosula, Shankar; Liu, Boli; Ding, Yu-Shin

25

Mapping the Target Localization and Biodistribution of Non-Radiolabeled VMAT2 Ligands in rat Brain

AAPS JOURNAL

2014, 16(3): 592-599

SCI

Deng, Aifang; Wu, Xianying; Zhou, Xue; Zhang, Yan; Yin, Wei; Qiao, Jinping; Zhu, Lin

26

Novel [(TcN)-Tc-99m](2+) Labeled EGFR Inhibitors as Potential Radiotracers for Single Photon Emission Computed Tomography (SPECT) Tumor Imaging

MOLECULES

2014, 19(5): 5508-5521

SCI

Zhao, Mingxia; Ning, Hongyu; Feng, Man; Li, Shilei; Chang, Jin; Qi, Chuanmin

27

Progressive loss of striatal dopamine terminals in MPTP-induced acute parkinsonism in cynomolgus monkeys using vesicular monoamine transporter type 2 PET imaging ([F-18]AV-133)

NEUROSCIENCE BULLETIN

2014, 30(3): 409-416

SCI

Liu, Yajing; Yue, Feng; Tang, Rongping; Tao, Guoxian; Pan, Xiaomei; Zhu, Lin; Kung, Hank F.; Chan, Piu

28

Radioiodinated Benzyloxybenzene Derivatives: A Class of Flexible Ligands Target to beta-Amyloid Plaques in Alzheimer's Brains

JOURNAL OF MEDICINAL CHEMISTRY

2014, 57(14): 6030-6042

SCI

Yang, Yanping; Cui, Mengchao; Zhang, Xiaoyang; Dai, Jiapei; Zhang, Zhiyong; Lin, Chunping; Guo, Yuzhi; Liu, Boli

29

Synthesis and biodistribution of Tc-99m-HYNIC-DG as a novel potential tumor imaging agent

NUCLEAR MEDICINE AND BIOLOGY

2014, 41(7): 622-623

SCI

Liu, Liqin; Zhao, Manchen; Wang, Zhuo; Qin, Yuanyan; Wang, Xuebin

30

Synthesis and preclinical evaluation of novel Pteroy-lys derivatives labeled with Tc-99m for FR-positive tumor imaging

NUCLEAR MEDICINE AND BIOLOGY

2014, 41(7): 627-628

SCI

Yu, Qian; Chen, Yuan; Zhang, Chun; He, Yingfang; Lu, Jie

31

A new kind of imaging agent for myocardial fatty acids metabolism

NUCLEAR MEDICINE AND BIOLOGY

2014, 41(7): 627

SCI

Xue, Tian; Li, Xiang; Liu, Jianping; Zhang, Huabei

32

Synthesis and biodistribution of (TcO)-Tc-99m-TRYDTC as a novel potential tumor imaging agent

NUCLEAR MEDICINE AND BIOLOGY

2014, 41(7): 621

SCI

Zhu, Jingjing; Hu, Qiran; Du, Jin; Wang, Xuebin; Zhang, Junbo

33

Synthesis and biodistribution of Tc-99m(CO)(3)-CPADG as a promising tumor imaging agent

NUCLEAR MEDICINE AND BIOLOGY

2014, 41(7): 621

SCI

Wang, Yue; Zhu, Jingjing; Song, Xiaoqing; Wang, Xuebin; Zhang, Junbo

34

GC法测定正电子类放射性药物制剂中有机溶剂残留量

解放军药学学报

2014, 30(4):

303-305

国内期刊

武仙英,贾娟娟,乔洪文,邓艾芳,乔晋萍,朱霖,钟建国

35

From bench to market: translational medicine in the development of

Molecular imaging agents

转化医学研究(电子版)

2014, 4(1): 21-31

国内期刊

Zhu Lin, Kung Hank F

36

多巴胺神经系统显像分子探针研究

生命的化学

2014, 02, 154-165

国内期刊

乔晋萍; 乔洪文; 武仙英; 邓艾芳; 朱霖

37

Synthesis and biodistribution of Tc-99m(CO)(3)-G12N3 as a potential agent for tumor imaging

NUCLEAR MEDICINE AND BIOLOGY

2014, 41(7): 621

SCI

Liu, Teli; Wang, Xuebin; Zhang, Junbo

38

Tc-99m(CO)(3)-labeled 2-phenylbenzothiazoles as A beta imaging agents for the detection of CAA

NUCLEAR MEDICINE AND BIOLOGY

2014, 41(7): 621

SCI

Jia, Jianhua; Cui, Mengchao; Liu, Boli

39

Synthesis and biological evaluation of (TcO)-Tc-99m-MNXT as a novel tumor hypoxia imaging agent

NUCLEAR MEDICINE AND BIOLOGY

2014, 41(7): 614

SCI

Li, Zhenxiang; Wang, Xuebin; Zhang, Junbo

40

[CpM(CO)(3)] (M = Re, Tc-99m) labeled phenylbenzothiazoles as imaging agents for A beta plaques

NUCLEAR MEDICINE AND BIOLOGY

2014, 41(7): 614

SCI

Jia, Jianhua; Cui, Mengchao; Liu, Bali

41

Kit formulated asialoglycoprotein receptor targeting tracer based on copolymer for liver SPECT imaging

NUCLEAR MEDICINE AND BIOLOGY

2014, 41(7): 587-593

SCI

Liu, Chang; Guo, Zhide; Zhang, Pu; Song, Manli; Zhao, Zuoquan; Wu, Xiaowei; Zhang, Xianzhong

42

Preparation and biodistribution of a Tc-99m tricarbonyl complex with deoxyglucose dithiocarbamate as a tumor imaging agent for SPECT

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

2014, 24(16): 3964-3967

SCI

Lin, Xiao; Chao, Xiaoyu; Zhang, Junbo; Jin, Zhonghui; Zhang, Yanyan

43

Synthesis and evaluation of Tc-99m-2-[(3-carboxy-1-oxopropyl)amino]-2-deoxy-D-glucose as a potential tumor imaging agent

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

2014, 24(16): 38823885

SCI

Wang, Yue; Zhu, Jingjing; Song, Xiaoqing; Wang, Xuebin; Yang, Jigang; Zhang, Junbo

44

An-jun-ning, a traditional herbal formula, attenuates spontaneous withdrawal symptoms via modulation of the dopamine system in morphine-dependent rats

BMC COMPLEMENTARY AND ALTERNATIVE MEDICINE

2014, 14, 308

SCI

Gao, Jin-Long; Tu, Shao-Ang; Liu, Jia; Zhang, Jin-Ming; Huang, Yiyun; Han, Mei; Liang, Jian-Hui

45

Novel Cyclopentadienyl Tricarbonyl Tc-99m Complexes Containing 1-Piperonylpiperazine Moiety: Potential Imaging Probes for Sigma-1 Receptors

JOURNAL OF MEDICINAL CHEMISTRY

2014, 57(16): 7113-7125

SCI

Wang, Xia; Li, Dan; Deuther-Conrad, Winnie; Lu, Jie; Xie, Ying; Jia, Bing; Cui, Mengchao; Steinbach, Joerg; Brust, Peter; Liu, Boli; Jia, Hongmei

46

Synthesis and preliminary evaluation of novel Tc-99m-labeled folate derivative via click reaction for SPECT imaging

APPLIED RADIATION AND ISOTOPES

2014, 91, 24-30

SCI

Guo, Zhide; Zhang, Pu; Song, Manli; Wu, Xiaowei; Liu, Chang; Zhao, Zuoquan; Lu, Jie; Zhang, Xianzhong

47

Synthesis and biological evaluation of novel technetium-99m-labeled HYNIC-D-glucose as a potential tumor imaging agent

JOURNAL OF RADIOANALYTICAL AND NUCLEAR CHEMISTRY

2014, 30(13): 731-737

SCI

Liu, Liqin; Zhao, Manchen; Wang, Zhuo; Qin, Yuanyan; Wang, Xuebin

48

Novel F-18-labeled dibenzylideneacetone derivatives as potential positron emission tomography probes for in vivo imaging of beta-amyloid plaques

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

2014, 84, 628-638

SCI

Li, Zijing; Cui, Mengchao; Zhang, Jinming; Dai, Jiapei; Zhang, Xiaojun; Chen, Peng; Jia, Hongmei; Liu, Boli

49

Synthesis and biological evaluation of novel Tc-99m-oxo and Tc-99m-nitrido complexes with phenylalanine dithiocarbamate for tumor imaging

JOURNAL OF RADIOANALYTICAL AND NUCLEAR CHEMISTRY

2014, 302(1): 211-216

SCI

Zhu, Jingjing; Wang, Yue; Li, Zhenxiang; Fang, Si'an; Zhang, Junbo

50

Synthesis and evaluation of a F-18-labeled spirocyclic piperidine derivative as promising sigma(1) receptor imaging agent

BIOORGANIC & MEDICINAL CHEMISTRY

2014, 22(19): 5270-5278

SCI

Chen, Yuan-Yuan; Wang, Xia; Zhang, Jin-Ming; Deuther-Conrad, Winnie; Zhang, Xiao-Jun; Huang, Yiyun; Li, Yan; Ye, Jia-Jun; Cui, Meng-Chao; Steinbach, Joerg; Brust, Peter; Liu, Bo-Li; Jia, Hong-Mei

51

Highly Efficient One-Pot Labeling of New Phosphonium Cations with Fluorine-18 as Potential PET Agents for Myocardial Perfusion Imaging

MOLECULAR PHARMACEUTICS

2014, 11(11): 3823-3831

SCI

Zhao, Zuoquan; Yu, Qian; Mou, Tiantian; Liu, Chang; Yang, Wenjiang; Fang, Wei; Peng, Cheng; Lu, Jie; Liu, Yu; Zhang, Xianzhong

52

Radiolabeled bioactive benzoheterocycles for imaging beta-amyloid plaques in Alzheimer's disease

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

2014, 87, 703-721

SCI

Yang, Yanping; Cui, Mengchao

 
 
2014年专利发表汇总
 

1

专利

-18标记的螺环哌啶类sigma-1受体化合物及制备方法和应用

贾红梅、李艳、张锦明、崔孟超、刘伯里

中国发明专利

ZL 2012 1 0097119.6.

2

专利

新型18F标记取代苯并咪唑类化合物及其制备方法和制备肿瘤PET显像剂中的应用

齐传民,王潇,张淑婷,贺勇,刘航,许荆立,李桂霞,冯曼

中国发明专利

200910157577.2

2014,06,4授权)

3

专利

新型18F标记间硝基苯甲酰基氨基酸、制备方法和在肿瘤显像剂中的应用

齐传民,乔雅丽,张淑婷,贺勇,刘航,李桂霞,许荆立

中国发明专利

200810167557.9

2014,04,16授权)

4

专利

新的18F取代对甲苯磺氧基标记的吡唑并[1,5-a]嘧啶类化合物及制备和应用

齐传民,刘航,李桂霞,贺勇,许荆立,丁瑞,张淑婷,王潇

中国发明专利

200910157360.1

2014,04,16授权)

5

专利

. 一种F-三唑环-聚乙二醇-2-硝基咪唑化合物及其制备方法.

朱霖; 杜风华; 刘亚静

中国发明专利

zl200910091132.9.2014.7.9.授权)

6

专利

18/19F-酯类硝基咪唑化合物及其制备方法和作为乏氧组织显像剂的用途.

朱霖,乔晋萍,杜晶磊.

中国发明专利

zl201210077912.X.2014.6.5授权)

7

专利

五羟色胺转运体显像剂[18F]-FPBM的标记方法.

朱霖,李根薰,李崧,乔晋萍..

中国发明专利

zl201110341561.4.2014.8.21. 授权)

8

专利

新型锝-99m标记的高级脂肪酸衍生物

张华北 曾华辉 于海静

中国发明专利

ZL201110149254.6 (授权2014.06.25授权)

 

9

专利

一种与斑块有亲和力的2-芳基苯并杂环化合物及其制备方法和应用

崔孟超 张锦明 王学丹 贾红梅 刘伯里

中国发明专利

201210135460.6

2014,12,31授权)

 

 


 

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